Dr Andrey Berezin
Postdoctoral Research Associate (with Prof Davide Bonifazi)
Publication
2024
- Williams, T. L. et al. 2024. Secondary amine catalysis in enzyme design: broadening protein template diversity through genetic code expansion. Angewandte Chemie International Edition (10.1002/anie.202403098)
2021
- Zhou, J. et al. 2021. Organic room-temperature phosphorescence from halogen-bonded organic frameworks: hidden electronic effects in rigidified chromophores. Chemical Science 12(2), pp. 767-773. (10.1039/D0SC04646A)
2018
- Sciutto, A., Berezin, A., Lo Cicero, M., Miletic, T., Stopin, A. and Bonifazi, D. 2018. Tailored synthesis of N-substituted peri-Xanthenoxanthene Diimide (PXXDI) and Monoimide (PXXMI) Scaffolds. Journal of Organic Chemistry 83(22), pp. 13787-13798. (10.1021/acs.joc.8b02076)
- Bonifazi, D., Berezin, A., Battisti, T. and Biot, N. 2018. Oxygen-doped zig-zag molecular ribbons. Angewandte Chemie - International Edition 57(29), pp. 8942-8946. (10.1002/anie.201803282)
- Keane, L. et al. 2018. Anti-cancer activity of Phenyl and Pyrid-2-yl 1,3-substituted Benzo[1,2,4]triazin-7-ones and stable free radical precursors. Molecules 23(3), article number: 574. (10.3390/molecules23030574)
2017
- Royer, J., Berezin, A. and Marinelli, D. 2017. Tert-butylation of naphthalene-2,6-diol and 6-methoxynaphthalen-2-ol. ARKIVOC 2017(3), pp. 287-292. (10.24820/ark.5550190.p010.242)
- Savva, A. C. et al. 2017. Preparation of Blatter radicals via aza-Wittig chemistry: The reaction of N-aryliminophosphoranes with 1-(het)aroyl-2-aryldiazenes. Journal of Organic Chemistry 82(14), pp. 7564-7575. (10.1021/acs.joc.7b01297)
2016
- Sweeney, M. et al. 2016. Discovery of anti-cancer activity for benzo[1,2,4]triazin-7-ones: Very strong correlation to pleurotin and thioredoxin reductase inhibition. Bioorganic and Medicinal Chemistry 24(16), pp. 3565-3570. (10.1016/j.bmc.2016.05.066)
- Constantinides, C., Berezin, A., Zissimou, G., Manoli, M., Leitus, G. and Koutentis, P. 2016. The suppression of Columnar π-Stacking in 3-Adamantyl-1-phenyl-1,4-dihydrobenzo[e][1,2,4]triazin-4-yl. Molecules 21(5), article number: 636. (10.3390/molecules21050636)
2015
- Rocard, L., Berezin, A., De Leo, F. and Bonifazi, D. 2015. Templated chromophore assembly by dynamic covalent bonds. Angewandte Chemie International Edition 54(52), pp. 15739-15743. (10.1002/anie.201507186)
- Constantinides, C. P. et al. 2015. Tetraphenylhexaazaanthracenes: 16π weakly antiaromatic species with singlet ground states. Organic Letters 17(16), pp. 4026-4029. (10.1021/acs.orglett.5b01923)
- Berezin, A., Sciutto, A., Demitri, N. and Bonifazi, D. 2015. Rational synthesis of AB-type N-substituted core-functionalized naphthalene diimides (cNDIs). Organic Letters 17(8), pp. 1870-1873. (10.1021/acs.orglett.5b00543)
2014
- Constantinides, C. P. et al. 2014. A Magnetostructural Investigation of an Abrupt Spin Transition for 1-Phenyl-3-trifluoromethyl-1,4-dihydrobenzo[e][1,2,4]triazin-4-yl. Journal of the American Chemical Society 136(34), pp. 11906-11909. (10.1021/ja5063746)
- Constantinides, C. P. et al. 2014. Structural, magnetic, and computational correlations of some imidazolo-fused 1,2,4-benzotriazinyl radicals. Chemistry - A European Journal 20(18), pp. 5388-5396. (10.1002/chem.201304538)
- Berezin, A. A. and Koutentis, P. A. 2014. Ring contraction of 1,3-diphenylbenzo[1,2,4]triazinyl radicals to 1,2-diphenylbenzimidazoles. Organic and Biomolecular Chemistry 12(10), pp. 1641-1648. (10.1039/C3OB42130A)
- Demetriou, M., Berezin, A. A., Koutentis, P. A. and Krasia-Christoforou, T. 2014. Benzotriazinyl-mediated controlled radical polymerization of styrene. Polymer International 63(4), pp. 674-679. (10.1002/pi.4566)
- Constantinides, C. P., Berezin, A. A., Manoli, M., Leitus, G. M., Bendikov, M., Rawson, J. M. and Koutentis, P. A. 2014. Effective exchange coupling in alternating-chains of a π-extended 1,2,4-benzotriazin-4-yl. New Journal of Chemistry 38(3), pp. 949-954. (10.1039/C3NJ01235B)
- Berezin, A. A., Zissimou, G., Constantinides, C. P., Beldjoudi, Y., Rawson, J. M. and Koutentis, P. A. 2014. Route to benzo- and pyrido-fused 1,2,4-triazinyl radicals via N′-(het)aryl-N′-[2-nitro(het)aryl]hydrazides. Journal of Organic Chemistry 79(1), pp. 314-327. (10.1021/jo402481t)
2013
- Berezin, A. A., Constantinides, C. P., Mirallai, S. I., Manoli, M., Cao, L. L., Rawson, J. M. and Koutentis, P. A. 2013. Synthesis and properties of imidazolo-fused benzotriazinyl radicals. Organic and Biomolecular Chemistry 11(39), pp. 6780-6864. (10.1039/c3ob41169a)
2012
- Catto, M. et al. 2012. Design, synthesis and biological evaluation of benzo[e][1,2,4]triazin-7(1H)-one and [1,2,4]-triazino[5,6,1-jk]carbazol-6-one derivatives as dual inhibitors of beta-amyloid aggregation and acetyl/butyryl cholinesterase. European Journal of Medicinal Chemistry 58, pp. 84-97. (10.1016/j.ejmech.2012.10.003)
- Berezin, A. A., Constantinides, C. P., Drouza, C., Manoli, M. and Koutentis, P. A. 2012. From Blatter Radical to 7-Substituted 1,3-Diphenyl-1,4-dihydrothiazolo[5′,4′:4,5]benzo[1,2-e][1,2,4]triazin-4-yls: Toward Multifunctional Materials. Organic Letters 14(21), pp. 5586-5589. (10.1021/ol302714j)
2011
- Berezin, A. A., Koutentis, P. A. and Manos, M. J. 2011. Synthesis of sulfur containing analogues of the soluble guanylate cyclase inhibitor 8-bromo-4H-[1,2,4]oxadiazolo[3,4-c][1,4]benzoxazin-1-one NS2028. Tetrahedron 67(30), pp. 5437-5443. (10.1016/j.tet.2011.05.071)
- Berezin, A. A. and Koutentis, P. A. 2011. Suzuki–Miyaura reactions of the soluble guanylate cyclase inhibitor NS2028: a non-product specific route to C-8 substituted analogues. Tetrahedron 67(22), pp. 4069-4078. (10.1016/j.tet.2011.04.003)
- Berezin, A. A. and Koutentis, P. A. 2011. 8-[2-Chloro-5-(trifluoromethyl)phenyl]-4H-[1,2,4]oxadiazolo-[3,4-c][1,4]benzoxazin-1-one. Molbank 2011(2), pp. -., article number: M728. (10.3390/M728)
2007
- Konstantinova, L. S., Berezin, A. A., Lysov, K. A. and Rakitin, O. A. 2007. Selective synthesis of bis[1,2]dithiolo[1,4]thiazines from 4-isopropylamino-5-chloro-1,2-dithiole-3-ones. Tetrahedron Letters 48(33), pp. 5851-5854. (10.1016/j.tetlet.2007.06.071)
- Konstantinova, L. S., Berezin, A. A. and Rakitin, O. A. 2007. Transformations of N-ethylamines into amide derivatives under the action of sulfur monochloride. Russian Chemical Bulletin 56(6), pp. 1178-1183. (10.1007/s11172-007-0179-9)
2006
- Konstantinova, L. S., Berezin, A. A., Lysov, K. A. and Rakitin, O. A. 2006. Synthesis of 5-mercapto-1,2-dithiole-3-thiones and their transformation into 5-chloro-1,2-dithiol-3-ones. Russian Chemical Bulletin 55(1), pp. 147-151. (10.1007/s11172-006-0228-9)
Articles
- Williams, T. L. et al. 2024. Secondary amine catalysis in enzyme design: broadening protein template diversity through genetic code expansion. Angewandte Chemie International Edition (10.1002/anie.202403098)
- Zhou, J. et al. 2021. Organic room-temperature phosphorescence from halogen-bonded organic frameworks: hidden electronic effects in rigidified chromophores. Chemical Science 12(2), pp. 767-773. (10.1039/D0SC04646A)
- Sciutto, A., Berezin, A., Lo Cicero, M., Miletic, T., Stopin, A. and Bonifazi, D. 2018. Tailored synthesis of N-substituted peri-Xanthenoxanthene Diimide (PXXDI) and Monoimide (PXXMI) Scaffolds. Journal of Organic Chemistry 83(22), pp. 13787-13798. (10.1021/acs.joc.8b02076)
- Bonifazi, D., Berezin, A., Battisti, T. and Biot, N. 2018. Oxygen-doped zig-zag molecular ribbons. Angewandte Chemie - International Edition 57(29), pp. 8942-8946. (10.1002/anie.201803282)
- Keane, L. et al. 2018. Anti-cancer activity of Phenyl and Pyrid-2-yl 1,3-substituted Benzo[1,2,4]triazin-7-ones and stable free radical precursors. Molecules 23(3), article number: 574. (10.3390/molecules23030574)
- Royer, J., Berezin, A. and Marinelli, D. 2017. Tert-butylation of naphthalene-2,6-diol and 6-methoxynaphthalen-2-ol. ARKIVOC 2017(3), pp. 287-292. (10.24820/ark.5550190.p010.242)
- Savva, A. C. et al. 2017. Preparation of Blatter radicals via aza-Wittig chemistry: The reaction of N-aryliminophosphoranes with 1-(het)aroyl-2-aryldiazenes. Journal of Organic Chemistry 82(14), pp. 7564-7575. (10.1021/acs.joc.7b01297)
- Sweeney, M. et al. 2016. Discovery of anti-cancer activity for benzo[1,2,4]triazin-7-ones: Very strong correlation to pleurotin and thioredoxin reductase inhibition. Bioorganic and Medicinal Chemistry 24(16), pp. 3565-3570. (10.1016/j.bmc.2016.05.066)
- Constantinides, C., Berezin, A., Zissimou, G., Manoli, M., Leitus, G. and Koutentis, P. 2016. The suppression of Columnar π-Stacking in 3-Adamantyl-1-phenyl-1,4-dihydrobenzo[e][1,2,4]triazin-4-yl. Molecules 21(5), article number: 636. (10.3390/molecules21050636)
- Rocard, L., Berezin, A., De Leo, F. and Bonifazi, D. 2015. Templated chromophore assembly by dynamic covalent bonds. Angewandte Chemie International Edition 54(52), pp. 15739-15743. (10.1002/anie.201507186)
- Constantinides, C. P. et al. 2015. Tetraphenylhexaazaanthracenes: 16π weakly antiaromatic species with singlet ground states. Organic Letters 17(16), pp. 4026-4029. (10.1021/acs.orglett.5b01923)
- Berezin, A., Sciutto, A., Demitri, N. and Bonifazi, D. 2015. Rational synthesis of AB-type N-substituted core-functionalized naphthalene diimides (cNDIs). Organic Letters 17(8), pp. 1870-1873. (10.1021/acs.orglett.5b00543)
- Constantinides, C. P. et al. 2014. A Magnetostructural Investigation of an Abrupt Spin Transition for 1-Phenyl-3-trifluoromethyl-1,4-dihydrobenzo[e][1,2,4]triazin-4-yl. Journal of the American Chemical Society 136(34), pp. 11906-11909. (10.1021/ja5063746)
- Constantinides, C. P. et al. 2014. Structural, magnetic, and computational correlations of some imidazolo-fused 1,2,4-benzotriazinyl radicals. Chemistry - A European Journal 20(18), pp. 5388-5396. (10.1002/chem.201304538)
- Berezin, A. A. and Koutentis, P. A. 2014. Ring contraction of 1,3-diphenylbenzo[1,2,4]triazinyl radicals to 1,2-diphenylbenzimidazoles. Organic and Biomolecular Chemistry 12(10), pp. 1641-1648. (10.1039/C3OB42130A)
- Demetriou, M., Berezin, A. A., Koutentis, P. A. and Krasia-Christoforou, T. 2014. Benzotriazinyl-mediated controlled radical polymerization of styrene. Polymer International 63(4), pp. 674-679. (10.1002/pi.4566)
- Constantinides, C. P., Berezin, A. A., Manoli, M., Leitus, G. M., Bendikov, M., Rawson, J. M. and Koutentis, P. A. 2014. Effective exchange coupling in alternating-chains of a π-extended 1,2,4-benzotriazin-4-yl. New Journal of Chemistry 38(3), pp. 949-954. (10.1039/C3NJ01235B)
- Berezin, A. A., Zissimou, G., Constantinides, C. P., Beldjoudi, Y., Rawson, J. M. and Koutentis, P. A. 2014. Route to benzo- and pyrido-fused 1,2,4-triazinyl radicals via N′-(het)aryl-N′-[2-nitro(het)aryl]hydrazides. Journal of Organic Chemistry 79(1), pp. 314-327. (10.1021/jo402481t)
- Berezin, A. A., Constantinides, C. P., Mirallai, S. I., Manoli, M., Cao, L. L., Rawson, J. M. and Koutentis, P. A. 2013. Synthesis and properties of imidazolo-fused benzotriazinyl radicals. Organic and Biomolecular Chemistry 11(39), pp. 6780-6864. (10.1039/c3ob41169a)
- Catto, M. et al. 2012. Design, synthesis and biological evaluation of benzo[e][1,2,4]triazin-7(1H)-one and [1,2,4]-triazino[5,6,1-jk]carbazol-6-one derivatives as dual inhibitors of beta-amyloid aggregation and acetyl/butyryl cholinesterase. European Journal of Medicinal Chemistry 58, pp. 84-97. (10.1016/j.ejmech.2012.10.003)
- Berezin, A. A., Constantinides, C. P., Drouza, C., Manoli, M. and Koutentis, P. A. 2012. From Blatter Radical to 7-Substituted 1,3-Diphenyl-1,4-dihydrothiazolo[5′,4′:4,5]benzo[1,2-e][1,2,4]triazin-4-yls: Toward Multifunctional Materials. Organic Letters 14(21), pp. 5586-5589. (10.1021/ol302714j)
- Berezin, A. A., Koutentis, P. A. and Manos, M. J. 2011. Synthesis of sulfur containing analogues of the soluble guanylate cyclase inhibitor 8-bromo-4H-[1,2,4]oxadiazolo[3,4-c][1,4]benzoxazin-1-one NS2028. Tetrahedron 67(30), pp. 5437-5443. (10.1016/j.tet.2011.05.071)
- Berezin, A. A. and Koutentis, P. A. 2011. Suzuki–Miyaura reactions of the soluble guanylate cyclase inhibitor NS2028: a non-product specific route to C-8 substituted analogues. Tetrahedron 67(22), pp. 4069-4078. (10.1016/j.tet.2011.04.003)
- Berezin, A. A. and Koutentis, P. A. 2011. 8-[2-Chloro-5-(trifluoromethyl)phenyl]-4H-[1,2,4]oxadiazolo-[3,4-c][1,4]benzoxazin-1-one. Molbank 2011(2), pp. -., article number: M728. (10.3390/M728)
- Konstantinova, L. S., Berezin, A. A., Lysov, K. A. and Rakitin, O. A. 2007. Selective synthesis of bis[1,2]dithiolo[1,4]thiazines from 4-isopropylamino-5-chloro-1,2-dithiole-3-ones. Tetrahedron Letters 48(33), pp. 5851-5854. (10.1016/j.tetlet.2007.06.071)
- Konstantinova, L. S., Berezin, A. A. and Rakitin, O. A. 2007. Transformations of N-ethylamines into amide derivatives under the action of sulfur monochloride. Russian Chemical Bulletin 56(6), pp. 1178-1183. (10.1007/s11172-007-0179-9)
- Konstantinova, L. S., Berezin, A. A., Lysov, K. A. and Rakitin, O. A. 2006. Synthesis of 5-mercapto-1,2-dithiole-3-thiones and their transformation into 5-chloro-1,2-dithiol-3-ones. Russian Chemical Bulletin 55(1), pp. 147-151. (10.1007/s11172-006-0228-9)